Phosphorhydrazides as urease and acetylcholinesterase inhibitors: biological evaluation and QSAR study
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چکیده
منابع مشابه
Synthesis and biological evaluation of thiophene derivatives as acetylcholinesterase inhibitors.
A series of new thiophene derivatives has been synthesized using the Gewald protocol. The acetylcholinesterase inhibition activity was assayed according to Ellman's method using donepezil as reference. Some of the compounds were found to be more potent inhibitors than the reference. 2-(2-(4-(4-Methoxyphenyl)piperazin-1-yl)acetamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxamide (IIId) showe...
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ژورنال
عنوان ژورنال: Journal of the Iranian Chemical Society
سال: 2016
ISSN: 1735-207X,1735-2428
DOI: 10.1007/s13738-016-0836-8